Title : 4-(Methylnitrosamino)-1-(3-pyridyl)-1-butanone-Induced Histone Acetylation via α7nAChR-Mediated PI3K/Akt Activation and Its Impact on γ-H2AX Generation.

Pub. Date : 2021 Dec 20

PMID : 34784199






2 Functional Relationships(s)
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1 Phosphoinositide-3-kinase (PI3K)/Akt inhibitors, LY294002, wortmannin, and GSK690693, also suppressed both Ac-H3 and gamma-H2AX, whereas KU-55933, an inhibitor of ataxia telangiectasia mutated (ATM) upstream of gamma-H2AX, inhibited gamma-H2AX but not Ac-H3. gamma-h2ax phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit gamma Homo sapiens
2 Phosphoinositide-3-kinase (PI3K)/Akt inhibitors, LY294002, wortmannin, and GSK690693, also suppressed both Ac-H3 and gamma-H2AX, whereas KU-55933, an inhibitor of ataxia telangiectasia mutated (ATM) upstream of gamma-H2AX, inhibited gamma-H2AX but not Ac-H3. gamma-h2ax phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit gamma Homo sapiens