Title : UGT1A1 and UGT1A3 activity and inhibition in human liver and intestinal microsomes and a recombinant UGT system under similar assay conditions using selective substrates and inhibitors.

Pub. Date : 2021 Nov

PMID : 34698602






1 Functional Relationships(s)
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Compound Name
Protein Name
Organism
1 UGT1A1 catalyzed beta-estradiol 3-beta-D-glucuronide formation showed allosteric sigmoidal kinetics in all enzyme systems; while UGT1A3 catalyzed CDCA 24-acyl-beta-D-glucuronide formation exhibited Michaelis-Menten kinetics in HLM, substrate inhibition kinetics in HIM and rUGT systems. 24-acyl-beta-d-glucuronide UDP glucuronosyltransferase family 1 member A3 Homo sapiens