Title : Discovery of First-in-Class Peptidomimetic Neurolysin Activators Possessing Enhanced Brain Penetration and Stability.

Pub. Date : 2021 Sep 9

PMID : 34436882






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1 Herein, we report the discovery and hit-to-lead optimization of first-in-class Nln activators based on histidine-containing dipeptide hits identified from a virtual screen. Dipeptides neurolysin (metallopeptidase M3 family) Mus musculus