Title : Ligand-Independent G Protein-Coupled Estrogen Receptor/G Protein-Coupled Receptor 30 Activity: Lack of Receptor-Dependent Effects of G-1 and 17β-Estradiol.

Pub. Date : 2021 Sep

PMID : 34330822






7 Functional Relationships(s)
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Sentence
Compound Name
Protein Name
Organism
1 GPR30 is a membrane receptor reported to bind 17beta-estradiol (E2) and mediate rapid non-genomic estrogen responses, hence also named G protein-coupled estrogen receptor (GPER). Estradiol G protein-coupled estrogen receptor 1 Homo sapiens
2 GPR30 is a membrane receptor reported to bind 17beta-estradiol (E2) and mediate rapid non-genomic estrogen responses, hence also named G protein-coupled estrogen receptor (GPER). Estradiol G protein-coupled estrogen receptor 1 Homo sapiens
3 GPR30 is a membrane receptor reported to bind 17beta-estradiol (E2) and mediate rapid non-genomic estrogen responses, hence also named G protein-coupled estrogen receptor (GPER). Estradiol G protein-coupled estrogen receptor 1 Homo sapiens
4 GPR30 is a membrane receptor reported to bind 17beta-estradiol (E2) and mediate rapid non-genomic estrogen responses, hence also named G protein-coupled estrogen receptor (GPER). Estradiol G protein-coupled estrogen receptor 1 Homo sapiens
5 GPR30 is a membrane receptor reported to bind 17beta-estradiol (E2) and mediate rapid non-genomic estrogen responses, hence also named G protein-coupled estrogen receptor (GPER). Estradiol G protein-coupled estrogen receptor 1 Homo sapiens
6 GPR30 is a membrane receptor reported to bind 17beta-estradiol (E2) and mediate rapid non-genomic estrogen responses, hence also named G protein-coupled estrogen receptor (GPER). Estradiol G protein-coupled estrogen receptor 1 Homo sapiens
7 Significance Statement Much controversy surrounds E2 and G-1 as GPR30 agonists. Estradiol G protein-coupled estrogen receptor 1 Homo sapiens