Title : The tertiary oxime monoisonitrosoacetone penetrates the brain, reactivates inhibited acetylcholinesterase, and reduces mortality and morbidity following lethal sarin intoxication in guinea pigs.

Pub. Date : 2021 Mar 15

PMID : 33548273






2 Functional Relationships(s)
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Compound Name
Protein Name
Organism
1 However, available oxime antidote 2-PAM only reactivates OP-inhibited AChE in peripheral tissues. Oximes acetylcholinesterase Cavia porcellus
2 Monoisonitrosoacetone (MINA), a tertiary oxime, reportedly reactivates AChE in the central nervous system (CNS). Oximes acetylcholinesterase Cavia porcellus