Title : Impairment of endoxifen formation in tamoxifen-treated premenopausal breast cancer patients carrying reduced-function CYP2D6 alleles.

Pub. Date : 2021 Mar

PMID : 32713032






2 Functional Relationships(s)
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1 Impairment of endoxifen formation in tamoxifen-treated premenopausal breast cancer patients carrying reduced-function CYP2D6 alleles. Tamoxifen cytochrome P450 family 2 subfamily D member 6 Homo sapiens
2 AIMS: Tamoxifen is bioactivated to endoxifen by polymorphic CYP2D6-dependent metabolism. Tamoxifen cytochrome P450 family 2 subfamily D member 6 Homo sapiens