Title : Bis(vinylsulfonyl)piperazines as efficient linkers for highly homogeneous antibody-drug conjugates.

Pub. Date : 2020 Mar 15

PMID : 32018094






2 Functional Relationships(s)
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1 We present bis(vinylsulfonyl)piperazines (BVP) as efficient linkers to selectively re-bridge disulfides at the antigen-binding fragment (Fab) regions and produce highly homogeneous conjugates with a loading of two drugs without disulfide scrambling. Disulfides FA complementation group B Homo sapiens
2 We present bis(vinylsulfonyl)piperazines (BVP) as efficient linkers to selectively re-bridge disulfides at the antigen-binding fragment (Fab) regions and produce highly homogeneous conjugates with a loading of two drugs without disulfide scrambling. Disulfides FA complementation group B Homo sapiens