Title : The inhibitory role of purinergic P2Y receptor on Mg2+ transport across intestinal epithelium-like Caco-2 monolayer.

Pub. Date : 2019 Jan

PMID : 30032468






4 Functional Relationships(s)
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1 An agonist of the P2Y2 receptor, but not the P2Y4 or P2Y6 receptor, suppressed Mg2+ transport across control and omeprazole-treated monolayers. Omeprazole purinergic receptor P2Y2 Homo sapiens
2 Omeprazole enhanced P2Y2 receptor expression in Caco-2 cells. Omeprazole purinergic receptor P2Y2 Homo sapiens
3 Forskolin and P2Y2 receptor agonist markedly enhanced apical HCO3- secretion by control and omeprazole-treated monolayers. Omeprazole purinergic receptor P2Y2 Homo sapiens
4 Antagonists of cystic fibrosis transmembrane conductance regulator (CFTR) and Na+-HCO3- cotransporter-1 (NBCe1) could nullify the inhibitory effect of P2Y2 receptor agonist on Mg2+ transport across control and omeprazole-treated Caco-2 monolayers. Omeprazole purinergic receptor P2Y2 Homo sapiens