Title : Rational Design and Synthesis of Modified Teixobactin Analogues: In Vitro Antibacterial Activity against Staphylococcus aureus, Propionibacterium acnes and Pseudomonas aeruginosa.

Pub. Date : 2018 Jun 26

PMID : 29741277






1 Functional Relationships(s)
Download
Sentence
Compound Name
Protein Name
Organism
1 Extensive antimicrobial susceptibility assessment against a panel of clinically relevant Staphylococcus aureus and Propionibacterium acnes strains led to the identification of the new lead compound, [Arg(Me)10 ,Nle11 ]teixobactin, with an excellent bactericidal activity (minimum inhibitory concentration (MIC)=2-4 mug mL-1 ). Arginine L1 cell adhesion molecule Mus musculus