Title : Inhibitory Effects of Danshen components on CYP2C8 and CYP2J2.

Pub. Date : 2018 Jun 1

PMID : 29689254






2 Functional Relationships(s)
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Sentence
Compound Name
Protein Name
Organism
1 Dihydrotanshinone I had moderate noncompetitive inhibition on CYP2J2 (Ki = 6.59 muM), but mechanism-based inhibition on CYP2C8 (KI = 0.43 muM, kinact = 0.097 min-1). dhts latexin Homo sapiens
2 Dihydrotanshinone I had moderate noncompetitive inhibition on CYP2J2 (Ki = 6.59 muM), but mechanism-based inhibition on CYP2C8 (KI = 0.43 muM, kinact = 0.097 min-1). dhts latexin Homo sapiens