Title : Identification and Structure-Function Study of Positive Allosteric Modulators of Kainate Receptors.

Pub. Date : 2017 Jun

PMID : 28360094






2 Functional Relationships(s)
Download
Sentence
Compound Name
Protein Name
Organism
1 4-cyclopropyl-7-fluoro-3,4-dihydro-2H-1,2,4-benzothiadiazine 1,1-dioxide (BPAM344) potentiated glutamate-evoked currents of GluK2a 21-fold at the highest concentration tested (200 muM), with an EC50 of 79 muM. Saccharin latexin Homo sapiens
2 4-cyclopropyl-7-fluoro-3,4-dihydro-2H-1,2,4-benzothiadiazine 1,1-dioxide (BPAM344) potentiated glutamate-evoked currents of GluK2a 21-fold at the highest concentration tested (200 muM), with an EC50 of 79 muM. Saccharin latexin Homo sapiens