Title : Bortezomib inhibits mammalian carbonic anhydrases.

Pub. Date : 2017 Oct 1

PMID : 28277280






1 Functional Relationships(s)
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1 The remaining cytosolic (CA III, VII and XIII), membrane-anchored (CA IV), mitochondrial (CA VA, VB), transmembrane (CA XII) and secreted (CA VI) isoforms were slightly less inhibited by bortezomib compared to isoforms discussed above, with KIs ranging between 4.38 and 8.45muM. Bortezomib carbonic anhydrase 5A Homo sapiens