Title : Nalfurafine is a G-protein biased agonist having significantly greater bias at the human than rodent form of the kappa opioid receptor.

Pub. Date : 2017 Apr

PMID : 28088389






1 Functional Relationships(s)
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1 Although nalfurafine is reported to have low receptor selectivity in radioligand binding assays, its antinociceptive effect was blocked by the selective KOR antagonist norbinaltorphimine. norbinaltorphimine opioid receptor kappa 1 Homo sapiens