Title : Attenuation of rifampicin-induced theophylline metabolism by diltiazem/rifampicin coadministration in healthy volunteers.

Pub. Date : 1989

PMID : 2792166






1 Functional Relationships(s)
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1 In these 6 volunteers, intake of diltiazem (240 mg daily), concurrently with rifampicin for a week, significantly elevated theophylline half-life to 6.2 h as well as reduced its clearance to 1.03 ml.min-1.kg-1. Diltiazem CD59 molecule (CD59 blood group) Homo sapiens