Title : Characterization of human cytochrome P450 mediated bioactivation of amodiaquine and its major metabolite N-desethylamodiaquine.

Pub. Date : 2017 Mar

PMID : 27718269






2 Functional Relationships(s)
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Protein Name
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1 For AQ bioactivation, enzyme kinetical parameters were Km , 11.5 +- 2.0 mumol l-1 , Vmax , 59.2 +- 3.2 pmol min-1 mg-1 and CLint , 5.15 mul min-1 mg-1 . Amodiaquine CD59 molecule (CD59 blood group) Homo sapiens
2 For AQ bioactivation, enzyme kinetical parameters were Km , 11.5 +- 2.0 mumol l-1 , Vmax , 59.2 +- 3.2 pmol min-1 mg-1 and CLint , 5.15 mul min-1 mg-1 . Amodiaquine CD59 molecule (CD59 blood group) Homo sapiens