Pub. Date : 2016 Sep 15
PMID : 27448773
2 Functional Relationships(s)Download |
Sentence | Compound Name | Protein Name | Organism |
1 | Steric structure-activity relationship of cyproheptadine derivatives as inhibitors of histone methyltransferase Set7/9. | Cyproheptadine | SET domain containing 7, histone lysine methyltransferase | Homo sapiens |
2 | We previously identified cyproheptadine, which has a characteristic butterfly-like molecular conformation with bent tricyclic dibenzosuberene and chair-form N-methylpiperidine moieties, as a Set7/9 inhibitor. | Cyproheptadine | SET domain containing 7, histone lysine methyltransferase | Homo sapiens |