Title : Expression of functional sphingosine-1 phosphate receptor-1 is reduced by B cell receptor signaling and increased by inhibition of PI3 kinase δ but not SYK or BTK in chronic lymphocytic leukemia cells.

Pub. Date : 2015 Mar 1

PMID : 25632006






1 Functional Relationships(s)
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1 BCR signaling pathway inhibitors such as ibrutinib, idelalisib, and fostamatinib (respective inhibitors of Bruton"s tyrosine kinase, PI3Kdelta, and spleen tyrosine kinase) represent a significant therapeutic advance in B cell malignancies, including chronic lymphocytic leukemia (CLL). idelalisib Bruton tyrosine kinase Homo sapiens