Title : Demethoxycurcumin modulates human P-glycoprotein function via uncompetitive inhibition of ATPase hydrolysis activity.

Pub. Date : 2015 Jan 28

PMID : 25594233






3 Functional Relationships(s)
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1 Demethoxycurcumin modulates human P-glycoprotein function via uncompetitive inhibition of ATPase hydrolysis activity. demethoxycurcumin dynein axonemal heavy chain 8 Homo sapiens
2 Demethoxycurcumin inhibited P-glycoprotein-mediated ATP hydrolysis under concentrations of <1 muM and efficiently inhibited 200 muM verapamil-stimulated ATPase activity, indicating a high affinity of demethoxycurcumin for P-glycoprotein. demethoxycurcumin dynein axonemal heavy chain 8 Homo sapiens
3 Demethoxycurcumin inhibited P-glycoprotein-mediated ATP hydrolysis under concentrations of <1 muM and efficiently inhibited 200 muM verapamil-stimulated ATPase activity, indicating a high affinity of demethoxycurcumin for P-glycoprotein. demethoxycurcumin dynein axonemal heavy chain 8 Homo sapiens