Title : Tricyclic antidepressants exhibit variable pharmacological profiles at the α(2A) adrenergic receptor.

Pub. Date : 2014 Aug 29

PMID : 25128275






1 Functional Relationships(s)
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1 Our previous work established a particular TCA, desipramine, as an arrestin-biased alpha2AAR ligand driving receptor endocytosis and downregulation but not canonical heterotrimeric G protein-mediated signaling. Desipramine adrenoceptor alpha 2A Homo sapiens