Title : Aminothiazole-featured pirinixic acid derivatives as dual 5-lipoxygenase and microsomal prostaglandin E2 synthase-1 inhibitors with improved potency and efficiency in vivo.

Pub. Date : 2013 Nov 27

PMID : 24171493






1 Functional Relationships(s)
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1 Together, 2-aminothiazole-featured pirinixic acids represent potent dual 5-LO/mPGES-1 inhibitors with an attractive pharmacological profile as anti-inflammatory drugs. 2-aminothiazole prostaglandin E synthase Mus musculus