Title : Activity, inhibition, and induction of cytochrome P450 2J2 in adult human primary cardiomyocytes.

Pub. Date : 2013 Dec

PMID : 24021950






1 Functional Relationships(s)
Download
Sentence
Compound Name
Protein Name
Organism
1 CYP2J2 activity in the cell line was inhibited by danazol, astemizole, and ketoconazole in submicromolar range, but also by xenobiotics known to cause cardiac adverse effects. Astemizole cytochrome P450 family 2 subfamily J member 2 Homo sapiens