Title : The HSP90 inhibitor 17-allylamino-17-demethoxygeldanamycin modulates radiosensitivity by downregulating serine/threonine kinase 38 via Sp1 inhibition.

Pub. Date : 2013 Nov

PMID : 23886587






1 Functional Relationships(s)
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1 The ansamycin-based HSP90 inhibitor 17-AAG (17-allylamino-17-demethoxygeldanamycin) combats tumors and has been shown to modulate cellular sensitivity to radiation, prompting researchers to use 17-AAG as a radiosensitizer. Rifabutin heat shock protein 90 alpha family class A member 1 Homo sapiens