Title : Largazole, a class I histone deacetylase inhibitor, enhances TNF-α-induced ICAM-1 and VCAM-1 expression in rheumatoid arthritis synovial fibroblasts.

Pub. Date : 2013 Jul 15

PMID : 23632129






1 Functional Relationships(s)
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1 Further, the addition of HDAC6 specific inhibitor Tubastatin A with LAR suppressed TNF-alpha+LAR-induced ICAM-1 and VCAM-1 expression and completely blocked MMP-2 activity, suggesting a role of HDAC6 in LAR-induced ICAM-1 and VCAM-1 expression. tubastatin A tumor necrosis factor Homo sapiens