Title : Chronic sazetidine-A at behaviorally active doses does not increase nicotinic cholinergic receptors in rodent brain.

Pub. Date : 2012 Nov

PMID : 22899752






1 Functional Relationships(s)
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1 We used a newly developed method involving radioligand binding to measure the concentrations and nAChR occupancy of saz-A, nicotine, and varenicline in brains from chronically treated rats. Varenicline cholinergic receptor nicotinic beta 1 subunit Rattus norvegicus