Title : N-(2-methyl-6-benzoxazolyl)-N'-1,5-naphthyridin-4-yl urea (SB334867), a hypocretin receptor-1 antagonist, preferentially prevents ethanol seeking: comparison with natural reward seeking.

Pub. Date : 2014 Mar

PMID : 22830647






2 Functional Relationships(s)
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1 N-(2-methyl-6-benzoxazolyl)-N"-1,5-naphthyridin-4-yl urea (SB334867), a hypocretin receptor-1 antagonist, preferentially prevents ethanol seeking: comparison with natural reward seeking. 1-(2-methylbenzoxazol-6-yl)-3-(1,5)naphthyridin-4-yl urea hypocretin receptor 1 Homo sapiens
2 This study was designed to test the effect of the specific Orx/Hcrt receptor-1 (Hcrt-r1) antagonist, N-(2-methyl-6-benzoxazolyl)-N"-1,5-naphthyridin-4-yl urea (SB334867), on reinstatement elicited by ethanol (EtOH)-associated stimuli versus stimuli associated with a conventional reinforcer [i.e. SuperSac, consisting of 3% glucose and 0.125% saccharin (w/v)]. 1-(2-methylbenzoxazol-6-yl)-3-(1,5)naphthyridin-4-yl urea hypocretin receptor 1 Homo sapiens