Title : Heat shock factor-1 knockout induces multidrug resistance gene, MDR1b, and enhances P-glycoprotein (ABCB1)-based drug extrusion in the heart.

Pub. Date : 2012 Jun 5

PMID : 22615365






1 Functional Relationships(s)
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1 Moreover, application of the P-gp antagonist, verapamil, increased Dox loading in HSF-1(-/-) cardiomyocytes, deteriorated cardiac function in HSF-1(-/-) mice, and decreased survival. Verapamil phosphoglycolate phosphatase Mus musculus