Title : Structural features discriminate androgen receptor N/C terminal and coactivator interactions.

Pub. Date : 2012 Jan 30

PMID : 21664945






1 Functional Relationships(s)
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Protein Name
Organism
1 High affinity equilibrium androgen binding was retained by alanine substitution mutations at Tyr-739 in AR LBD helix 5 or Lys-905 in helix 12 structurally adjacent to AF2, whereas transcriptional activity decreased and the androgen dissociation increased. Alanine androgen receptor Homo sapiens