Title : Rimonabant is a dual inhibitor of acyl CoA:cholesterol acyltransferases 1 and 2.

Pub. Date : 2010 Aug 6

PMID : 20609360






2 Functional Relationships(s)
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1 Rimonabant inhibited ACAT activity in intact CHO-ACAT1 and CHO-ACAT2 cells and in cell-free assays with approximately equal efficiency (IC(50)=1.5+/-1.2 microM and 2.2+/-1.1 microM for CHO-ACAT1 and CHO-ACAT2, respectively). Rimonabant acetyl-CoA acetyltransferase 2 Homo sapiens
2 Rimonabant inhibited ACAT activity in intact CHO-ACAT1 and CHO-ACAT2 cells and in cell-free assays with approximately equal efficiency (IC(50)=1.5+/-1.2 microM and 2.2+/-1.1 microM for CHO-ACAT1 and CHO-ACAT2, respectively). Rimonabant acetyl-CoA acetyltransferase 2 Homo sapiens