Title : Trifluoromethylpyrimidine-based inhibitors of proline-rich tyrosine kinase 2 (PYK2): structure-activity relationships and strategies for the elimination of reactive metabolite formation.

Pub. Date : 2008 Dec 1

PMID : 18951788






1 Functional Relationships(s)
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1 The synthesis and SAR for a series of diaminopyrimidines as PYK2 inhibitors are described. diaminopyrimidines protein tyrosine kinase 2 beta Homo sapiens