Title : Design, synthesis and structure-activity relationship of simple bis-amides as potent inhibitors of GlyT1.

Pub. Date : 2008 Oct 15

PMID : 18805008






1 Functional Relationships(s)
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Protein Name
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1 Several novel classes of potent and small amide-type inhibitors of glycine transport (GlyT1) were developed through sequential simplification of a benzodiazepinone-lead structure identified from a high-throughput screening. Glycine solute carrier family 6 member 9 Homo sapiens