Title : Effects of human immunodeficiency virus protease inhibitors on the intestinal absorption of tenofovir disoproxil fumarate in vitro.

Pub. Date : 2007 Oct

PMID : 17664327






1 Functional Relationships(s)
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1 Pgp inhibition constants ranged from 10.3 microM (lopinavir) to >100 microM (amprenavir, indinavir, and darunavir). Lopinavir PGP Canis lupus familiaris