Title : From dihydroxypyrimidine carboxylic acids to carboxamide HIV-1 integrase inhibitors: SAR around the amide moiety.

Pub. Date : 2007 Jan 15

PMID : 17107799






1 Functional Relationships(s)
Download
Sentence
Compound Name
Protein Name
Organism
1 Extensive SAR around the benzylamide moiety led to the identification of the p-fluorobenzylamide as optimal in the enzymatic assay. beclamide sarcosine dehydrogenase Homo sapiens