Title : Guggulsterone activates multiple nuclear receptors and induces CYP3A gene expression through the pregnane X receptor.

Pub. Date : 2004 Aug

PMID : 15075359






2 Functional Relationships(s)
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1 Here, we show that guggulsterones activate the estrogen receptor alpha isoform, progesterone receptor, and pregnane X receptor. pregna-4,17-diene-3,16-dione estrogen receptor 1 Homo sapiens
2 Moreover, our data suggest the need for additional studies of guggulsterones agonist activity against estrogen receptor alpha isoform and the progesterone receptor. pregna-4,17-diene-3,16-dione estrogen receptor 1 Homo sapiens