Title : Effects of the EGFR/HER2 kinase inhibitor GW572016 on EGFR- and HER2-overexpressing breast cancer cell line proliferation, radiosensitization, and resistance.

Pub. Date : 2004 Feb 1

PMID : 14751502






1 Functional Relationships(s)
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1 Exploration of potential mechanisms of resistance in SUM185 cells revealed failure of GW572016 to inhibit downstream ERK and Akt activation, despite inhibition of HER2 phosphorylation. Lapatinib AKT serine/threonine kinase 1 Homo sapiens