Title : Novel CFTR chloride channel activators identified by screening of combinatorial libraries based on flavone and benzoquinolizinium lead compounds.

Pub. Date : 2001 Jun 8

PMID : 11262417






3 Functional Relationships(s)
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Compound Name
Protein Name
Organism
1 The flavonoid genistein and the benzo[c]quinolizinium MPB-07 have been shown to activate the cystic fibrosis transmembrane conductance regulator (CFTR), the protein that is defective in cystic fibrosis. Genistein CF transmembrane conductance regulator Homo sapiens
2 The flavonoid genistein and the benzo[c]quinolizinium MPB-07 have been shown to activate the cystic fibrosis transmembrane conductance regulator (CFTR), the protein that is defective in cystic fibrosis. Genistein CF transmembrane conductance regulator Homo sapiens
3 Compared with genistein, the most active compounds had up to 10 times greater potency in activating wild-type and/or G551D-CFTR. Genistein CF transmembrane conductance regulator Homo sapiens