MLN 8237


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83 Functionally related protein(s)
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Protein Name
UniProt Entry
Gene Symbol
Organism
NCBI Gene ID
# All related compound(s)
#Article(s)
1 aurora kinase A AURKA_HUMAN AURKA Homo sapiens 6790 433 110
2 aurora kinase A AURKA_MOUSE Aurka Mus musculus 20878 82 15
3 AKT serine/threonine kinase 1 AKT1_HUMAN AKT1 Homo sapiens 207 6445 9
4 tumor protein p53 P53_HUMAN TP53 Homo sapiens 7157 5584 8
5 mechanistic target of rapamycin kinase MTOR_HUMAN MTOR Homo sapiens 2475 3411 6
6 mitogen-activated protein kinase 14 MK14_HUMAN MAPK14 Homo sapiens 1432 3132 5
7 MYC proto-oncogene, bHLH transcription factor MYC_HUMAN MYC Homo sapiens 4609 2261 4
8 ATP binding cassette subfamily B member 1 MDR1_HUMAN ABCB1 Homo sapiens 5243 3985 3
9 MYCN proto-oncogene, bHLH transcription factor MYCN_HUMAN MYCN Homo sapiens 4613 374 3
10 cytochrome P450 family 3 subfamily A member 4 CP3A4_HUMAN CYP3A4 Homo sapiens 1576 3475 3
11 cyclin D1 CCND1_HUMAN CCND1 Homo sapiens 595 1747 2
12 poly(ADP-ribose) polymerase 1 PARP1_HUMAN PARP1 Homo sapiens 142 2571 2
13 BH3 interacting domain death agonist BID_HUMAN BID Homo sapiens 637 1130 2
14 transformation related protein 53, pseudogene - Trp53-ps Mus musculus 22060 1552 2
15 myelocytomatosis oncogene MYC_MOUSE Myc Mus musculus 17869 289 2
16 BCL2 apoptosis regulator BCL2_HUMAN BCL2 Homo sapiens 596 4403 2
17 enhancer of zeste 2 polycomb repressive complex 2 subunit EZH2_HUMAN EZH2 Homo sapiens 2146 470 2
18 v-myc avian myelocytomatosis viral related oncogene, neuroblastoma derived MYCN_MOUSE Mycn Mus musculus 18109 102 2
19 nuclear paraspeckle assembly transcript 1 - NEAT1 Homo sapiens 283131 176 1
20 RAS like proto-oncogene A RALA_HUMAN RALA Homo sapiens 5898 186 1
21 cadherin 1 CADH1_HUMAN CDH1 Homo sapiens 999 1360 1
22 annexin A5 ANXA5_HUMAN ANXA5 Homo sapiens 308 1785 1
23 cytochrome P450 family 2 subfamily D member 6 CP2D6_HUMAN CYP2D6 Homo sapiens 1565 1531 1
24 CD38 molecule CD38_HUMAN CD38 Homo sapiens 952 501 1
25 O-6-methylguanine-DNA methyltransferase MGMT_HUMAN MGMT Homo sapiens 4255 549 1
26 polycystin 2, transient receptor potential cation channel PKD2_MOUSE Pkd2 Mus musculus 18764 88 1
27 translocated promoter region, nuclear basket protein TPR_HUMAN TPR Homo sapiens 7175 238 1
28 triosephosphate isomerase 1 TPIS_HUMAN TPI1 Homo sapiens 7167 355 1
29 cytochrome P450 family 2 subfamily C member 19 CP2CJ_HUMAN CYP2C19 Homo sapiens 1557 1098 1
30 cytochrome P450 family 2 subfamily C member 9 CP2C9_HUMAN CYP2C9 Homo sapiens 1559 1244 1
31 thymoma viral proto-oncogene 1 AKT1_MOUSE Akt1 Mus musculus 11651 3034 1
32 MCL1 apoptosis regulator, BCL2 family member MCL1_HUMAN MCL1 Homo sapiens 4170 1015 1
33 BRCA2 DNA repair associated BRCA2_HUMAN BRCA2 Homo sapiens 675 305 1
34 phosphoglycolate phosphatase PGP_MOUSE Pgp Mus musculus 67078 756 1
35 cytochrome P450 family 2 subfamily C member 8 CP2C8_HUMAN CYP2C8 Homo sapiens 1558 590 1
36 polo like kinase 1 PLK1_HUMAN PLK1 Homo sapiens 5347 475 1
37 von Hippel-Lindau tumor suppressor VHL_HUMAN VHL Homo sapiens 7428 215 1
38 ATM serine/threonine kinase ATM_HUMAN ATM Homo sapiens 472 847 1
39 sirtuin 1 SIR1_HUMAN SIRT1 Homo sapiens 23411 1253 1
40 ATP binding cassette subfamily C member 1 MRP1_HUMAN ABCC1 Homo sapiens 4363 1125 1
41 ATP binding cassette subfamily G member 2 (Junior blood group) ABCG2_HUMAN ABCG2 Homo sapiens 9429 1370 1
42 tumor protein p73 P73_HUMAN TP73 Homo sapiens 7161 217 1
43 transformation related protein 53 P53_MOUSE Trp53 Mus musculus 22059 281 1
44 catenin beta 1 CTNB1_HUMAN CTNNB1 Homo sapiens 1499 2350 1
45 ribosomal protein S6 kinase B1 KS6B1_HUMAN RPS6KB1 Homo sapiens 6198 764 1
46 CD274 molecule PD1L1_HUMAN CD274 Homo sapiens 29126 1115 1
47 B cell leukemia/lymphoma 2 BCL2_MOUSE Bcl2 Mus musculus 12043 1497 1
48 DNA methyltransferase 1 DNMT1_HUMAN DNMT1 Homo sapiens 1786 621 1
49 mitogen-activated protein kinase 3 MK03_MOUSE Mapk3 Mus musculus 26417 1527 1
50 cyclin dependent kinase 4 CDK4_HUMAN CDK4 Homo sapiens 1019 868 1