Propafenone

ATP binding cassette subfamily B member 1 ; Homo sapiens







15 Article(s)
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1 31917466 Propafenone analogue with additional H-bond acceptor group shows increased inhibitory activity on P-glycoprotein. 2020 Mar 2
2 26970257 Subtle Structural Differences Trigger Inhibitory Activity of Propafenone Analogues at the Two Polyspecific ABC Transporters: P-Glycoprotein (P-gp) and Breast Cancer Resistance Protein (BCRP). 2016 Jun 20 2
3 22452412 Structure-activity relationships, ligand efficiency, and lipophilic efficiency profiles of benzophenone-type inhibitors of the multidrug transporter P-glycoprotein. 2012 Apr 12 2
4 21177413 Molecular dissection of dual pseudosymmetric solute translocation pathways in human P-glycoprotein. 2011 Mar 1
5 21589945 Exhaustive sampling of docking poses reveals binding hypotheses for propafenone type inhibitors of P-glycoprotein. 2011 May 3
6 18303146 Venlafaxine-propafenone interaction resulting in hallucinations and psychomotor agitation. 2008 Mar 1
7 16843673 Studies of interactions between uracil-based hybrid molecules and P-glycoprotein--search for multidrug resistance modulators. 2006 Nov 1 2
8 15900513 Characterisation of (R/S)-propafenone and its metabolites as substrates and inhibitors of P-glycoprotein. 2005 Mar 5
9 16082413 Targeting drug-efflux pumps -- a pharmacoinformatic approach. 2005 3
10 16787327 Interaction field based and hologram based QSAR analysis of propafenone-type modulators of multidrug resistance. 2005 Sep 1
11 15188222 Intramolecular distribution of hydrophobicity influences pharmacological activity of propafenone-type MDR modulators. 2004 Jun 1
12 11854445 Identification of ligand-binding regions of P-glycoprotein by activated-pharmacophore photoaffinity labeling and matrix-assisted laser desorption/ionization-time-of-flight mass spectrometry. 2002 Mar 1
13 12825790 Similarity based SAR (SIBAR) as tool for early ADME profiling. 2002 Nov 1
14 10513988 Structure-activity relationship studies of propafenone analogs based on P-glycoprotein ATPase activity measurements. 1999 Nov 1 3
15 9747179 A combined Hansch/Free-Wilson approach as predictive tool in QSAR studies on propafenone-type modulators of multidrug resistance. 1998 Jul-Aug 1