GSK5182

estrogen related receptor gamma ; Homo sapiens







16 Article(s)
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Pub. Year
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1 33612148 The estrogen-related receptor γ modulator, GSK5182, inhibits osteoclast differentiation and accelerates osteoclast apoptosis. 2021 May 6
2 32079653 Estrogen-related receptors are targetable ROS sensors. 2020 Apr 1 1
3 32173553 Regulation of dopaminergic neuronal phenotypes by the estrogen-related receptor gamma ligand GSK4716 via the activation of CREB signaling. 2020 Jun 1
4 31479733 Estrogen-related receptor γ controls sterol regulatory element-binding protein-1c expression and alcoholic fatty liver. 2019 Dec 1
5 30019168 Inverse agonist of ERRγ reduces cannabinoid receptor type 1-mediated induction of fibrinogen synthesis in mice with a high-fat diet-intoxicated liver. 2018 Sep 1
6 28382164 Visualization of Macrophage Recruitment to Inflammation Lesions using Highly Sensitive and Stable Radionuclide-Embedded Gold Nanoparticles as a Nuclear Bio-Imaging Platform. 2017 1
7 28750085 Orphan nuclear receptor ERRγ is a key regulator of human fibrinogen gene expression. 2017 1
8 26771593 Identification of Selective ERRγ Inverse Agonists. 2016 Jan 12 2
9 26940882 Estrogen-related receptor γ is upregulated in liver cancer and its inhibition suppresses liver cancer cell proliferation via induction of p21 and p27. 2016 Mar 4 1
10 27236015 Synthesis and biological evaluation of novel 4-hydroxytamoxifen analogs as estrogen-related receptor gamma inverse agonists. 2016 Sep 14 1
11 25451157 In vitro metabolism of an estrogen-related receptor γ modulator, GSK5182, by human liver microsomes and recombinant cytochrome P450s. 2015 Apr 3
12 26338896 Inverse Agonist of Estrogen-Related Receptor γ Enhances Sodium Iodide Symporter Function Through Mitogen-Activated Protein Kinase Signaling in Anaplastic Thyroid Cancer Cells. 2015 Nov 2
13 24466039 Orphan nuclear receptor Errγ induces C-reactive protein gene expression through induction of ER-bound Bzip transmembrane transcription factor CREBH. 2014 1
14 23050013 Hypoxia induces PDK4 gene expression through induction of the orphan nuclear receptor ERRγ. 2012 1
15 21911493 Estrogen-related receptor γ (ERRγ) is a novel transcriptional regulator of phosphatidic acid phosphatase, LIPIN1, and inhibits hepatic insulin signaling. 2011 Nov 4 1
16 19690166 Transcriptional corepressor SMILE recruits SIRT1 to inhibit nuclear receptor estrogen receptor-related receptor gamma transactivation. 2009 Oct 16 4