PMID-sentid Pub_year Sent_text comp_official_name comp_offsetprotein_name organism prot_offset 25471566-2 2014 Whereas Thio-THIP displayed weak antagonist activity at alpha1,2,5beta2,3gamma2S and rho1 GABAARs and partial agonism at alpha6beta2,3delta GABAARs expressed in Xenopus oocytes, the pronounced agonism exhibited by the compound at alpha4beta1delta and alpha4beta3delta GABAARs was contrasted by its negligible activity at the alpha4beta2delta subtype. Thio-THIP 8-17 MGC75582, possible similarity to act2 S homeolog Xenopus laevis 56-71