PMID-sentid Pub_year Sent_text comp_official_name comp_offsetprotein_name organism prot_offset 23586323-4 2013 EXPERIMENTAL APPROACH: hERG and K(IR)2.1 trafficking in HEK293 cells was evaluated by Western blot and immunofluorescence microscopy after treatment with pentamidine and six pentamidine analogues, and correction with dofetilide and four dofetilide analogues that displayed different abilities to inhibit IKr . Pentamidine 154-165 ETS transcription factor ERG Homo sapiens 23-27 23586323-4 2013 EXPERIMENTAL APPROACH: hERG and K(IR)2.1 trafficking in HEK293 cells was evaluated by Western blot and immunofluorescence microscopy after treatment with pentamidine and six pentamidine analogues, and correction with dofetilide and four dofetilide analogues that displayed different abilities to inhibit IKr . Pentamidine 174-185 ETS transcription factor ERG Homo sapiens 23-27 23586323-6 2013 KEY RESULTS: Structural modifications of pentamidine differentially affected plasma membrane levels of hERG and K(IR)2.1. Pentamidine 41-52 ETS transcription factor ERG Homo sapiens 103-107 23586323-9 2013 Dofetilide corrected pentamidine-induced hERG, but not K(IR)2.1 trafficking defects. Pentamidine 21-32 ETS transcription factor ERG Homo sapiens 41-45