PMID-sentid	Pub_year	Sent_text	compound_name	comp_offset	prot_official_name	organism	prot_offset
20066493-1	2011	The apical sodium-codependent bile acid transporter (ASBT) inhibition activity of benzothiepine derivatives have been analyzed based on topological and molecular features.	1-Benzothiepin	82-95	solute carrier family 10 member 2	Homo sapiens	53-57
16134950-6	2005	The reported results describe the synthesis and SAR development of this benzothiepine class of ASBT inhibitors resulting in an 6000-fold improvement in ASBT inhibition with desired minimal systemic exposure of this locally acting drug candidate.	1-Benzothiepin	72-85	solute carrier family 10 member 2	Homo sapiens	95-99
16134950-6	2005	The reported results describe the synthesis and SAR development of this benzothiepine class of ASBT inhibitors resulting in an 6000-fold improvement in ASBT inhibition with desired minimal systemic exposure of this locally acting drug candidate.	1-Benzothiepin	72-85	solute carrier family 10 member 2	Homo sapiens	152-156
16134951-4	2005	A series of benzothiepines were prepared to refine the structure-activity relationship of the substituted phenyl ring at the 5-position of benzothiepine ring and to identify potent, crystalline, nonhygroscopic, and efficacious ASBT inhibitors with low systemic exposure.	1-Benzothiepin	12-25	solute carrier family 10 member 2	Homo sapiens	227-231