PMID-sentid Pub_year Sent_text compound_name comp_offset prot_official_name organism prot_offset 27066749-4 2016 These insights allowed for the design of GSK2807, a potent and selective, SAM-competitive inhibitor of SMYD3 (Ki = 14 nM). GSK2807 41-48 SET and MYND domain containing 3 Homo sapiens 103-108 27066749-5 2016 A high-resolution crystal structure reveals that GSK2807 bridges the gap between the SAM-binding pocket and the substrate lysine tunnel of SMYD3. GSK2807 49-56 SET and MYND domain containing 3 Homo sapiens 139-144