PMID-sentid Pub_year Sent_text comp_official_name comp_offsetprotein_name organism prot_offset 28094183-0 2017 Discovering novel 7-azaindole-based series as potent AXL kinase inhibitors. 7-azaindole dimer 18-29 AXL receptor tyrosine kinase Homo sapiens 53-56 28094183-3 2017 In this context, we started to design new kinase inhibitors targeting AXL from the 7-azaindole scaffold well known to interact with the ATP binding site of the kinase. 7-azaindole dimer 83-94 AXL receptor tyrosine kinase Homo sapiens 70-73 28094183-4 2017 Focused screening and chemical diversification around 7-azaindole scaffold were developed, based on modeling studies and medicinal chemistry rational, leading to the discovery of a new family of hits with potent inhibitory activity against AXL. 7-azaindole dimer 54-65 AXL receptor tyrosine kinase Homo sapiens 240-243