PMID-sentid	Pub_year	Sent_text		comp_official_name	comp_offsetprotein_name	organism	prot_offset
33612148-5	2021	Interestingly, GSK5182 increased ERRgamma protein levels much as does GSK4716, which is an ERRgamma agonist.	GSK 4716	70-77	estrogen related receptor gamma	Homo sapiens	91-99	
16990259-7	2006	The observed agonist-bound state contains the ERRgamma LBD, a ligand (GSK4716), and the RIP140 peptide and reveals an unexpected rearrangement of the phenol-binding residues.	GSK 4716	70-77	estrogen related receptor gamma	Homo sapiens	46-54	
16990259-9	2006	In contrast to the conventional mechanism of nuclear receptor ligand activation, activation of ERRgamma by GSK4716 does not appear to involve a major rearrangement or significant stabilization of the C-terminal helix.	GSK 4716	107-114	estrogen related receptor gamma	Homo sapiens	95-103	
32897058-5	2020	Here, we describe a novel dual ERRalpha/gamma inverse agonist, SLU-PP-1072, derived from the GSK4716 ERRgamma agonist scaffold that is distinct from the XCT790 scaffold.	GSK 4716	93-100	estrogen related receptor gamma	Homo sapiens	101-109	
32173553-0	2020	Regulation of dopaminergic neuronal phenotypes by the estrogen-related receptor gamma ligand GSK4716 via the activation of CREB signaling.	GSK 4716	93-100	estrogen related receptor gamma	Homo sapiens	54-85	
31491697-5	2019	All of the tested chemicals could bind to ERRgamma with the Kd (dissociation constant) values ranging from not available (NA) to 3.2 muM 4"-OH-PCB 12 showed the highest binding affinity with Kd value of 3.2 muM, which was comparable to that of a synthetic ERRgamma agonist GSK4716.	GSK 4716	273-280	estrogen related receptor gamma	Homo sapiens	42-50	
16515477-7	2006	The phenolic acyl hydrazones GSK4716 and GSK9089 act as selective agonists of ERRbeta and ERRgamma.	GSK 4716	29-36	estrogen related receptor gamma	Homo sapiens	90-98	
15857113-2	2005	GSK4716 (3) and GSK9089 (4) show binding to ERRgamma with remarkable selectivity over the classical estrogen receptors.	GSK 4716	0-7	estrogen related receptor gamma	Homo sapiens	44-52