PMID-sentid	Pub_year	Sent_text		comp_official_name	comp_offsetprotein_name	organism	prot_offset
31097402-5	2019	Thereby, oxime derivatives with a 1,1"-biphenyl moiety were found as the first inhibitors of mGAT1 comprising a pyrrolidine-3-carboxylic acid motif with affinities in the submicromolar range.	Oximes	9-14	solute carrier family 6 (neurotransmitter transporter, GABA), member 1	Mus musculus	93-98	
30777661-1	2019	Generation and screening of oxime libraries by competitive MS Binding Assays represents a powerful tool for the identification of new compounds, with affinity to mGAT1, the most abundant plasma membrane bound GABA transporter in the CNS.	Oximes	28-33	solute carrier family 6 (neurotransmitter transporter, GABA), member 1	Mus musculus	162-167	
30777661-2	2019	By screening a guvacine derived oxime library, new potent inhibitors of mGAT1 had been revealed.	Oximes	32-37	solute carrier family 6 (neurotransmitter transporter, GABA), member 1	Mus musculus	72-77	
30777661-3	2019	In the present study, oxime libraries generated by reaction of a large excess of a rac-nipecotic acid derivative displaying a hydroxylamine functionality in which various aldehydes under suitable conditions, were examined for new potent inhibitors of mGAT1.	Oximes	22-27	solute carrier family 6 (neurotransmitter transporter, GABA), member 1	Mus musculus	251-256	
30485691-1	2018	In this study, pyrrolidine-3-acetic acid derived oxime libraries were applied to the concept of library screening by MS Binding Assays, as a powerful technique to reveal new potent murine gamma-aminobutyric acid transporter subtype (mGAT1) inhibitors.	Oximes	49-54	solute carrier family 6 (neurotransmitter transporter, GABA), member 1	Mus musculus	233-238	
30485691-3	2018	The oxime libraries have been screened by means of competitive MS Binding Assays and, as a consequence, the most active libraries were further investigated through deconvolution experiments to identify single oximes responsible for the observed activity on the target mGAT1.	Oximes	4-9	solute carrier family 6 (neurotransmitter transporter, GABA), member 1	Mus musculus	268-273	
30485691-3	2018	The oxime libraries have been screened by means of competitive MS Binding Assays and, as a consequence, the most active libraries were further investigated through deconvolution experiments to identify single oximes responsible for the observed activity on the target mGAT1.	Oximes	209-215	solute carrier family 6 (neurotransmitter transporter, GABA), member 1	Mus musculus	268-273