PMID-sentid Pub_year Sent_text comp_official_name comp_offsetprotein_name organism prot_offset 34298950-4 2021 In this study, we identified pyridine derivatives by evaluating in vitro TNKS enzyme activity and investigated N-((1,2,4)triazolo(4,3-a)pyridin-3-yl)-1-(2-cyanophenyl)piperidine-4-carboxamide (TI-12403) as a novel TNKS inhibitor. pyridine 29-37 tankyrase Homo sapiens 73-77 34298950-4 2021 In this study, we identified pyridine derivatives by evaluating in vitro TNKS enzyme activity and investigated N-((1,2,4)triazolo(4,3-a)pyridin-3-yl)-1-(2-cyanophenyl)piperidine-4-carboxamide (TI-12403) as a novel TNKS inhibitor. pyridine 29-37 tankyrase Homo sapiens 214-218