Title : Synthetic G protein-coupled bile acid receptor agonists and bile acids act via basolateral receptors in ileal and colonic mucosa.

Pub. Date : 2020 Dec

PMID : 32656959






5 Functional Relationships(s)
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Protein Name
Organism
1 Luminal TDCA crossed the epithelial lining via the apical sodium-dependent BA transporter (ASBT) and its inhibitor, GSK2330672 significantly reduced luminal, but not basolateral TDCA activity. Phenobarbital solute carrier family 10 member 2 Homo sapiens
2 Luminal TDCA crossed the epithelial lining via the apical sodium-dependent BA transporter (ASBT) and its inhibitor, GSK2330672 significantly reduced luminal, but not basolateral TDCA activity. Phenobarbital solute carrier family 10 member 2 Homo sapiens
3 Luminal TDCA crossed the epithelial lining via the apical sodium-dependent BA transporter (ASBT) and its inhibitor, GSK2330672 significantly reduced luminal, but not basolateral TDCA activity. Phenobarbital solute carrier family 10 member 2 Homo sapiens
4 Luminal TDCA crossed the epithelial lining via the apical sodium-dependent BA transporter (ASBT) and its inhibitor, GSK2330672 significantly reduced luminal, but not basolateral TDCA activity. Phenobarbital solute carrier family 10 member 2 Homo sapiens
5 Furthermore, luminal-conjugated BAs require transport across the epithelium via ASBT in order to activate basolateral GPBA. Phenobarbital solute carrier family 10 member 2 Homo sapiens