| 1 |
35565470 | P-glycoprotein Mediates Resistance to the Anaplastic Lymphoma Kinase Inhiitor Ensartinib in Cancer Cells. | 2022 May 9 |
1 |
| 2 |
33189788 | Novel dendritic polyglycerol-conjugated, mesoporous silica-based targeting nanocarriers for co-delivery of doxorubicin and tariquidar to overcome multidrug resistance in breast cancer stem cells. | 2021 Feb 10 |
3 |
| 3 |
33315404 | Pharmacokinetic Modeling of (R)-[11C]verapamil to Measure the P-Glycoprotein Function in Nonhuman Primates. | 2021 Jan 4 |
1 |
| 4 |
33838147 | Structural Basis of Drug Recognition by the Multidrug Transporter ABCG2. | 2021 Jun 25 |
3 |
| 5 |
33860196 | Inhibition of P-Glycoprotein Does Not Increase the Efficacy of Proteasome Inhibitors in Multiple Myeloma Cells. | 2021 Apr 9 |
1 |
| 6 |
33901197 | Transport of Alzheimer's associated amyloid-β catalyzed by P-glycoprotein. | 2021 |
2 |
| 7 |
33929088 | Computer-Aided Search for 5-Arylideneimidazolone Anticancer Agents Able To Overcome ABCB1-Based Multidrug Resistance. | 2021 Aug 5 |
1 |
| 8 |
34084427 | Active participation of membrane lipids in inhibition of multidrug transporter P-glycoprotein. | 2021 Apr 9 |
1 |
| 9 |
34208283 | The Long-Term DEHP Exposure Confers Multidrug Resistance of Triple-Negative Breast Cancer Cells through ABC Transporters and Intracellular ROS. | 2021 Jun 11 |
1 |
| 10 |
34220523 | ABCB1 and ABCG2 Together Limit the Distribution of ABCB1/ABCG2 Substrates to the Human Retina and the ABCG2 Single Nucleotide Polymorphism Q141K (c.421C> A) May Lead to Increased Drug Exposure. | 2021 |
5 |
| 11 |
34617531 | A multidrug-resistant P-glycoprotein assembly revealed by tariquidar-probe's super-resolution imaging. | 2021 Oct 21 |
1 |
| 12 |
32056006 | Restoration of MARCKS enhances chemosensitivity in cancer. | 2020 Apr |
1 |
| 13 |
32176509 | Folic Acid-Modified Nanoerythrocyte for Codelivery of Paclitaxel and Tariquidar to Overcome Breast Cancer Multidrug Resistance. | 2020 Apr 6 |
1 |
| 14 |
32253945 | 6,7-Dimethoxy-2-phenethyl-1,2,3,4-tetrahydroisoquinoline amides and corresponding ester isosteres as multidrug resistance reversers. | 2020 Dec |
2 |
| 15 |
32256321 | Cannabidiol (CBD) Inhibited Rhodamine-123 Efflux in Cultured Vascular Endothelial Cells and Astrocytes Under Hypoxic Conditions. | 2020 |
1 |
| 16 |
32331368 | Insights into P-Glycoprotein Inhibitors: New Inducers of Immunogenic Cell Death. | 2020 Apr 22 |
2 |
| 17 |
32634436 | Overexpression of ABCB1 and ABCG2 contributes to reduced efficacy of the PI3K/mTOR inhibitor samotolisib (LY3023414) in cancer cell lines. | 2020 Oct |
1 |
| 18 |
30237210 | A Proof-of-Concept Study to Inhibit ABCG2- and ABCB1-Mediated Efflux Transport at the Human Blood-Brain Barrier. | 2019 Apr |
1 |
| 19 |
30391800 | Human iPSC-derived blood-brain barrier microvessels: validation of barrier function and endothelial cell behavior. | 2019 Jan |
1 |
| 20 |
31048454 | Coexpression of ABCB1 and ABCG2 in a Cell Line Model Reveals Both Independent and Additive Transporter Function. | 2019 Jul |
1 |
| 21 |
31379495 | Convulsive Stress Mimics Brain Hypoxia and Promotes the P-Glycoprotein (P-gp) and Erythropoietin Receptor Overexpression. Recombinant Human Erythropoietin Effect on P-gp Activity. | 2019 |
1 |
| 22 |
31441108 | Discovery to solve multidrug resistance: Design, synthesis, and biological evaluation of novel agents. | 2019 Oct |
1 |
| 23 |
31515284 | A High-Throughput Screen of a Library of Therapeutics Identifies Cytotoxic Substrates of P-glycoprotein. | 2019 Nov |
1 |
| 24 |
31774117 | ATP-dependent thermostabilization of human P-glycoprotein (ABCB1) is blocked by modulators. | 2019 Dec 19 |
1 |
| 25 |
31832814 | Assessment of brain delivery of a model ABCB1/ABCG2 substrate in patients with non-contrast-enhancing brain tumors with positron emission tomography. | 2019 Dec 12 |
2 |
| 26 |
29377455 | LysoTracker and MitoTracker Red are transport substrates of P-glycoprotein: implications for anticancer drug design evading multidrug resistance. | 2018 Apr |
1 |
| 27 |
29631786 | Design, synthesis and biological evaluation of novel tetrahydroisoquinoline derivatives as P-glycoprotein-mediated multidrug resistance inhibitors. | 2018 May 15 |
1 |
| 28 |
30041718 | Folate-Targeted Redox-Responsive Polymersomes Loaded with Chemotherapeutic Drugs and Tariquidar to Overcome Drug Resistance. | 2018 Oct 1 |
1 |
| 29 |
30453546 | Androgen Receptor Splice Variant 7 Drives the Growth of Castration Resistant Prostate Cancer without Being Involved in the Efficacy of Taxane Chemotherapy. | 2018 Nov 16 |
3 |
| 30 |
30562739 | Inhibition of Cyclin D1 Expression in Human Glioblastoma Cells is Associated with Increased Temozolomide Chemosensitivity. | 2018 |
1 |
| 31 |
27738009 | Assessment of P-Glycoprotein Transport Activity at the Human Blood-Retina Barrier with (R)-11C-Verapamil PET. | 2017 Apr |
1 |
| 32 |
28189725 | Role of P-glycoprotein inhibitors in ceramide-based therapeutics for treatment of cancer. | 2017 Apr 15 |
1 |
| 33 |
28509582 | Tariquidar sensitizes multiple myeloma cells to proteasome inhibitors via reduction of hypoxia-induced P-gp-mediated drug resistance. | 2017 Dec |
3 |
| 34 |
26622052 | Using the BacMam Baculovirus System to Study Expression and Function of Recombinant Efflux Drug Transporters in Polarized Epithelial Cell Monolayers. | 2016 Feb |
2 |
| 35 |
26913287 | 3D-QSAR AND CONTOUR MAP ANALYSIS OF TARIQUIDAR ANALOGUES AS MULTIDRUG RESISTANCE PROTEIN-1 (MRP1) INHIBITORS. | 2016 Feb |
1 |
| 36 |
26989076 | β-casein nanovehicles for oral delivery of chemotherapeutic Drug combinations overcoming P-glycoprotein-mediated multidrug resistance in human gastric cancer cells. | 2016 Apr 26 |
1 |
| 37 |
27522191 | Intracellular accumulation of Praziquantel in T lymphoblastoid cell lines, CEM (parental) and CEMVBL(P-gp-overexpressing). | 2016 Aug 14 |
1 |
| 38 |
27676469 | Phenyltetrazolyl-phenylamides: Substituent impact on modulation capability and selectivity toward the efflux protein ABCG2 and investigation of interaction with the transporter. | 2016 Nov 29 |
1 |
| 39 |
25669913 | Approaching complete inhibition of P-glycoprotein at the human blood-brain barrier: an (R)-[11C]verapamil PET study. | 2015 May |
2 |
| 40 |
25855895 | HM30181 Derivatives as Novel Potent and Selective Inhibitors of the Breast Cancer Resistance Protein (BCRP/ABCG2). | 2015 May 14 |
1 |
| 41 |
26125482 | Multiple Drug Transport Pathways through Human P-Glycoprotein. | 2015 Jul 21 |
1 |
| 42 |
26202880 | Factors Governing P-Glycoprotein-Mediated Drug-Drug Interactions at the Blood-Brain Barrier Measured with Positron Emission Tomography. | 2015 Sep 8 |
2 |
| 43 |
26486517 | Pharmacokinetic and pharmacodynamic study of tariquidar (XR9576), a P-glycoprotein inhibitor, in combination with doxorubicin, vinorelbine, or docetaxel in children and adolescents with refractory solid tumors. | 2015 Dec |
2 |
| 44 |
26507655 | Mapping the Binding Site of the Inhibitor Tariquidar That Stabilizes the First Transmembrane Domain of P-glycoprotein. | 2015 Dec 4 |
3 |
| 45 |
24478983 | Small and Innovative Molecules as New Strategy to Revert MDR. | 2014 |
1 |
| 46 |
25330312 | Inhibition or knockdown of ABC transporters enhances susceptibility of adult and juvenile schistosomes to Praziquantel. | 2014 Oct |
1 |
| 47 |
25456855 | Tariquidar inhibits P-glycoprotein drug efflux but activates ATPase activity by blocking transition to an open conformation. | 2014 Dec 15 |
4 |
| 48 |
23063413 | Establishment of a robust hepatitis C virus replicon cell line over-expressing P-glycoprotein that facilitates analysis of P-gp drug transporter effects on inhibitor antiviral activity. | 2013 Jan 1 |
1 |
| 49 |
23146816 | Pharmacokinetics of single ascending doses of the P-glycoprotein inhibitor tariquidar in healthy subjects. | 2013 |
3 |
| 50 |
23340958 | Retrospective analysis of P-glycoprotein-mediated drug-drug interactions at the blood-brain barrier in humans. | 2013 Apr |
1 |