Raloxifene Hydrochloride

estrogen receptor 2 ; Homo sapiens







33 Article(s)
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1 30615483 Raloxifene nano-micelles effect on triple-negative breast cancer is mediated through estrogen receptor-β and epidermal growth factor receptor. 2019 Sep 1
2 28003814 The Selective Estrogen Receptor Modulator Raloxifene Inhibits Neutrophil Extracellular Trap Formation. 2016 1
3 22398780 Estrogen receptor β potentiates the antiproliferative effect of raloxifene and affects the cell migration and invasion in HCT-116 colon cancer cells. 2012 Jul 2
4 22476901 The enhanced antiproliferative response to combined treatment of trichostatin A with raloxifene in MCF-7 breast cancer cells and its relevance to estrogen receptor β expression. 2012 Jul 4
5 20945400 Raloxifene induces cell death and inhibits proliferation through multiple signaling pathways in prostate cancer cells expressing different levels of estrogen receptor α and β. 2011 May 1
6 20659801 A mutant selective anti-estrogen is a pure antagonist on EREs and AP-1 response elements. 2010 Sep 1 1
7 19059307 Cell type- and estrogen receptor-subtype specific regulation of selective estrogen receptor modulator regulatory elements. 2009 Feb 27 3
8 19139018 Estrogen receptor-beta as a potential target for colon cancer prevention: chemoprevention of azoxymethane-induced colon carcinogenesis by raloxifene in F344 rats. 2009 Jan 1
9 17962382 Differential regulation of native estrogen receptor-regulatory elements by estradiol, tamoxifen, and raloxifene. 2008 Feb 2
10 18579664 Intratumoral estrogens and estrogen receptors in human non-small cell lung carcinoma. 2008 Jul 15 1
11 17135255 In vitro fluorescence anisotropy analysis of the interaction of full-length SRC1a with estrogen receptors alpha and beta supports an active displacement model for coregulator utilization. 2007 Feb 2 1
12 17336289 Raloxifene plus 17beta-estradiol inhibits proliferation of primary cultured vascular smooth muscle cells and human mammary endothelial cells via the janus kinase/signal transducer and activator of transcription3 cascade. 2007 Apr 30 1
13 17348852 Flexible estrogen receptor modulators: synthesis, biochemistry and molecular modeling studies for 3-benzyl-4,6-diarylhex-3-ene and 3,4,6-triarylhex-3-ene derivatives. 2007 Mar 1
14 16536755 Raloxifene, an oestrogen-receptor-beta-targeted therapy, inhibits androgen-independent prostate cancer growth: results from preclinical studies and a pilot phase II clinical trial. 2006 Apr 1
15 16554039 Evaluation of ligand selectivity using reporter cell lines stably expressing estrogen receptor alpha or beta. 2006 May 14 2
16 16700038 Expression of estrogen receptors-alpha and -beta in bladder cancer cell lines and human bladder tumor tissue. 2006 Jun 15 1
17 16787364 Antiestrogenically active 2-benzyl-1,1-diarylbut-2-enes: synthesis, structure-activity relationships and molecular modeling study for flexible estrogen receptor antagonists. 2006 Mar 1
18 16798746 Raloxifene increases proliferation and up-regulates telomerase activity in human umbilical vein endothelial cells. 2006 Aug 25 1
19 16010412 Potential of endogenous estrogen receptor beta to influence the selective ER modulator ERbeta complex. 2005 Aug 1
20 14699072 Estradiol and selective estrogen receptor modulators differentially regulate target genes with estrogen receptors alpha and beta. 2004 Mar 2
21 15138633 Differential effects of estradiol, raloxifene and tamoxifen on estrogen receptor expression in cultured human skin fibroblasts. 2004 Jun 2
22 12714703 Functional implications of antiestrogen induction of quinone reductase: inhibition of estrogen-induced deoxyribonucleic acid damage. 2003 Jul 1
23 14533013 Differential effects of estradiol and raloxifene on collagen biosynthesis in cultured human skin fibroblasts. 2003 Nov 1
24 11861516 Antagonists selective for estrogen receptor alpha. 2002 Mar 1
25 11060287 Unique protein determinants of the subtype-selective ligand responses of the estrogen receptors (ERalpha and ERbeta ) at AP-1 sites. 2001 Feb 9 1
26 11500849 Multiplexed molecular interactions of nuclear receptors using fluorescent microspheres. 2001 Aug 1 2
27 11720858 Activity of a tamoxifen-raloxifene hybrid ligand for estrogen receptors at an AP-1 site. 2001 Dec 17 2
28 10076999 Estrogen receptor beta activates the human retinoic acid receptor alpha-1 promoter in response to tamoxifen and other estrogen receptor antagonists, but not in response to estrogen. 1999 Mar 2
29 10395487 Estrogen receptor subtype-selective ligands: asymmetric synthesis and biological evaluation of cis- and trans-5,11-dialkyl- 5,6,11, 12-tetrahydrochrysenes. 1999 Jul 1 2
30 10469641 Structure of the ligand-binding domain of oestrogen receptor beta in the presence of a partial agonist and a full antagonist. 1999 Sep 1 1
31 9647865 Basic guide to the mechanisms of antiestrogen action. 1998 Jun 1
32 9658195 Differential response of estrogen receptor alpha and estrogen receptor beta to partial estrogen agonists/antagonists. 1998 Jul 1
33 9278514 Differential ligand activation of estrogen receptors ERalpha and ERbeta at AP1 sites. 1997 Sep 5 1