| 1 |
33054569 | Molecular networking based dereplication of AChE inhibitory compounds from the medicinal plant Vincetoxicum funebre (Boiss. & Kotschy). | 2022 Mar |
1 |
| 2 |
34971946 | Novel thiophene Chalcones-Coumarin as acetylcholinesterase inhibitors: Design, synthesis, biological evaluation, molecular docking, ADMET prediction and molecular dynamics simulation. | 2022 Feb |
1 |
| 3 |
35098414 | Alzheimer's disease therapy based on acetylcholinesterase inhibitor/blocker effects on voltage-gated potassium channels. | 2022 Mar |
2 |
| 4 |
35462270 | A single-molecule with multiple investigations: Synthesis, characterization, computational methods, inhibitory activity against Alzheimer's disease, toxicity, and ADME studies. | 2022 Apr 18 |
1 |
| 5 |
35527546 | A Cobalt-Containing Compound as a Stronger Inhibitor than Galantamine to Inhibit Acetylcholinesterase Activity: A New Drug Candidate for Alzheimer's Disease Treatment. | 2022 |
1 |
| 6 |
35563466 | Kinetic Modeling of Time-Dependent Enzyme Inhibition by Pre-Steady-State Analysis of Progress Curves: The Case Study of the Anti-Alzheimer's Drug Galantamine. | 2022 May 3 |
2 |
| 7 |
35595404 | Pharmacogenetic studies in Alzheimer disease. | 2022 May |
1 |
| 8 |
35630613 | Virtual Screening and Hit Selection of Natural Compounds as Acetylcholinesterase Inhibitors. | 2022 May 13 |
2 |
| 9 |
32146656 | Synthesis, biological evaluation, theoretical investigations, docking study and ADME parameters of some 1,4-bisphenylhydrazone derivatives as potent antioxidant agents and acetylcholinesterase inhibitors. | 2021 Feb |
1 |
| 10 |
33030113 | Multi-target approach for Alzheimer's disease treatment: computational biomolecular modeling of cholinesterase enzymes with a novel 4-N-phenylaminoquinoline derivative reveal promising potentials. | 2021 Jul |
1 |
| 11 |
33540879 | Anti-Cholinesterase Combination Drug Therapy as a Potential Treatment for Alzheimer's Disease. | 2021 Feb 2 |
1 |
| 12 |
33776997 | The Cholinergic Drug Galantamine Alleviates Oxidative Stress Alongside Anti-inflammatory and Cardio-Metabolic Effects in Subjects With the Metabolic Syndrome in a Randomized Trial. | 2021 |
1 |
| 13 |
33916760 | Discovery of a Novel Acetylcholinesterase Inhibitor by Fragment-Based Design and Virtual Screening. | 2021 Apr 3 |
1 |
| 14 |
34132933 | Machine learning models to select potential inhibitors of acetylcholinesterase activity from SistematX: a natural products database. | 2021 Aug |
1 |
| 15 |
34299650 | Bio-Guided Fractionation of Stem Bark Extracts from Phyllanthus muellarianus: Identification of Phytocomponents with Anti-Cholinesterase Activity. | 2021 Jul 20 |
1 |
| 16 |
34363318 | Structural Fractal Analysis of the Active Site of Acetylcholinesterase in Complexes with Huperzine A, Galantamine, and Donepezil. | 2021 Nov |
2 |
| 17 |
34443482 | Synthesis, Biological Evaluation, and In Silico Studies of New Acetylcholinesterase Inhibitors Based on Quinoxaline Scaffold. | 2021 Aug 12 |
1 |
| 18 |
34628223 | Synthesis, characterization, in vitro cholinesterase and hRBCs hemolysis assay and computational evaluation of novel 2,3,4,5-tetrahydrobenzothiazepine appended α-aminophosphonates. | 2021 Nov |
1 |
| 19 |
34664067 | UHPLC With On-Line Coupled Biochemical Detection for High Throughput Screening of Acetylcholinesterase Inhibitors in Coptidis Rhizoma and Cortex Phellodendri. | 2021 Oct 19 |
1 |
| 20 |
34755546 | Synthesis, molecular modeling and cholinesterase inhibitory effects of 2-indolinone-based hydrazinecarbothioamides. | 2021 Dec |
1 |
| 21 |
31686175 | Evidence for positive allosteric modulation of cognitive-enhancing effects of nicotine in healthy human subjects. | 2020 Jan |
2 |
| 22 |
31978679 | Design, synthesis and evaluation of pyrazole bearing α-aminophosphonate derivatives as potential acetylcholinesterase inhibitors against Alzheimer's disease. | 2020 Mar |
1 |
| 23 |
32414155 | Improving Anti-Neurodegenerative Benefits of Acetylcholinesterase Inhibitors in Alzheimer's Disease: Are Irreversible Inhibitors the Future? | 2020 May 13 |
1 |
| 24 |
32454229 | Simple analogues of natural product chelerythrine: Discovery of a novel anticholinesterase 2-phenylisoquinolin-2-ium scaffold with excellent potency against acetylcholinesterase. | 2020 Aug 15 |
1 |
| 25 |
32470371 | Highly potent cholinesterase inhibition of geranylated xanthones from Garcinia fusca and molecular docking studies. | 2020 Oct |
2 |
| 26 |
32717861 | Galantamine-Curcumin Hybrids as Dual-Site Binding Acetylcholinesterase Inhibitors. | 2020 Jul 23 |
3 |
| 27 |
32759369 | Oral Pretreatment with Galantamine Effectively Mitigates the Acute Toxicity of a Supralethal Dose of Soman in Cynomolgus Monkeys Posttreated with Conventional Antidotes. | 2020 Oct |
1 |
| 28 |
32763546 | Meta-analysis of randomized controlled trials of galantamine in schizophrenia: significant cognitive enhancement. | 2020 Sep |
1 |
| 29 |
32874532 | QT interval prolongation and Torsades de Pointes with donepezil, rivastigmine and galantamine. | 2020 |
1 |
| 30 |
33382027 | Revealing the cholinergic inhibition mechanism of Alzheimer's by galantamine: a metadynamics simulation study. | 2020 Dec 31 |
7 |
| 31 |
33488178 | Combined ligand and structure-based virtual screening approaches for identification of novel AChE inhibitors. | 2020 |
1 |
| 32 |
29697300 | Cooperative hydrogen bonds and mobility of the non-aromatic ring as selectivity determinants for human acetylcholinesterase to similar anti-Alzheimer's galantaminics: a computational study. | 2019 Apr |
2 |
| 33 |
30101703 | Phytoconstituents and their Possible Mechanistic Profile for Alzheimer's Disease - A Literature Review. | 2019 |
1 |
| 34 |
30673880 | Advances in Management of Psychosis in Neurodegenerative Diseases. | 2019 Jan 23 |
1 |
| 35 |
30819081 | Synthesis of New Galanthamine-Peptide Derivatives Designed for Prevention and Treatment of Alzheimer's Disease. | 2019 |
1 |
| 36 |
30956012 | Design, synthesis, evaluation and molecular modeling study of 4-N-phenylaminoquinolines for Alzheimer disease treatment. | 2019 Jun 1 |
1 |
| 37 |
31222828 | Novel fluorine-containing chiral hydrazide-hydrazones: Design, synthesis, structural elucidation, antioxidant and anticholinesterase activity, and in silico studies. | 2019 Aug |
1 |
| 38 |
31315114 | Effect of Rivastigmine (Acetyl Cholinesterase Inhibitor) versus Placebo on Manic Episodes in Patients with Bipolar Disorders: Results from a Double Blind, Randomized, Placebo-Controlled Clinical Trial. | 2019 |
1 |
| 39 |
31847089 | Synergistic Inhibition of Acetylcholinesterase by Alkaloids Derived from Stephaniae Tetrandrae Radix, Coptidis Rhizoma and Phellodendri Chinensis Cortex. | 2019 Dec 13 |
2 |
| 40 |
28974110 | Acetylcholinesterase Inhibitors: Beneficial Effects on Comorbidities in Patients With Alzheimer's Disease. | 2018 Mar |
1 |
| 41 |
29044771 | Alkaloids of Amaryllidaceae as Inhibitors of Cholinesterases (AChEs and BChEs): An Integrated Bioguided Study. | 2018 Mar |
1 |
| 42 |
29286595 | Galantamine and Computerized Cognitive Behavioral Therapy for Cocaine Dependence: A Randomized Clinical Trial. | 2018 Jan/Feb |
1 |
| 43 |
29570959 | Galantamine-Memantine Combination for Cognitive Impairments Due to Electroconvulsive Therapy, Traumatic Brain Injury, and Neurologic and Psychiatric Disorders: Kynurenic Acid and Mismatch Negativity Target Engagement. | 2018 Mar 1 |
1 |
| 44 |
29635172 | Combination of human acetylcholinesterase and serum albumin sensing surfaces as highly informative analytical tool for inhibitor screening. | 2018 Jun 5 |
1 |
| 45 |
29655025 | Design, facile synthesis, and evaluation of novel spiro- and pyrazolo[1,5-c]quinazolines as cholinesterase inhibitors: Molecular docking and MM/GBSA studies. | 2018 Jun |
1 |
| 46 |
29723743 | Spiropyrrolidine/spiroindolizino[6,7-b]indole heterocyclic hybrids: Stereoselective synthesis, cholinesterase inhibitory activity and their molecular docking study. | 2018 Sep |
1 |
| 47 |
29926988 | Effects of galantamine on smoking behavior and cognitive performance in treatment-seeking smokers prior to a quit attempt. | 2018 Jul |
1 |
| 48 |
30079554 | Synthesis, characterization, and SAR of arylated indenoquinoline-based cholinesterase and carbonic anhydrase inhibitors. | 2018 Sep |
1 |
| 49 |
30343499 | Thiazole-substituted benzoylpiperazine derivatives as acetylcholinesterase inhibitors. | 2018 Dec |
1 |
| 50 |
30643787 | Potential Role of Antipsychotic-Galantamine-Memantine Combination in the Treatment of Positive, Cognitive, and Negative Symptoms of Schizophrenia. | 2018 Dec |
1 |